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Oxycodone waxay ku jirtay isticmaalka kiliinikada ilaa 1917. Ka iibso Oxycodone Oxycontin 30mg online gudaha Australia
Waxa lagu maamulay bini'aadamka xididka (iv),
intramuscularly (im),
gudaha sanka (gudaha),
subka hoostiisa (sc),
si toos ah,
epidurally,
iyo afka iyadoo la isticmaalayo xalalka degdega ah, iyo kiniiniyada sii daynta degdega ah iyo kantaroolka. Iibso Oxycodone Oxycontin 30mg online gudaha Australia
Waddada ka gudubta maamulka ayaa sidoo kale lagu tijaabiyay xoolaha.
Taariikhda | Oxycontin ee Maareynta Xanuunka | Mushroomifi.
Waxa loo isticmaali jiray waqooyiga Yurub inta badan xanuunka ba'an. Kanada, Australia, iyo Maraykanka, waxaa inta badan loo isticmaali jiray daawo isku dhafan oo leh acetaminophen, phenacetin, iyo kafeyn loogu talagalay xanuunka dhexdhexaadka ah. Finland gudaheeda, oxycodone waxaa loo isticmaalay sidii opioid parenteral ugu weyn ee xanuunka ba'an tan iyo 1960-yadii. Iibso Oxycodone Oxycontin 30mg online gudaha Australia.
Kiimikada iyo Farmashiga aasaasiga ah | OxyContin 30 mg kaniiniyada sii daynta daba dheeraatay | Mushroomifi.
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Xidhiidhka xidhidhiyaha μ-opioid ee oxycodone, si kastaba ha ahaatee, wuu ka yar yahay kan morphine ama methadone.
Oxymorphone, dheef-shiid kiimikaadka firfircoon ee oxycodone, wuxuu leeyahay xidhiidh aad u sarreeya oo μ-opioid reseptor xidhidh.
Oxymorphone-ka intramuscular iyo morphine ayaa la barbardhigay bukaanada qaba xanuunka joogtada ah ee kansarka. Oxymorphone-ka muruqa dhexda ayaa 8.7 jeer ka awood badan morphine marka loo eego wadarta saamaynta xanuunka iyo 13 jeer marka la eego saamaynta ugu sarreysa.
Daraasadaha dabeecadda ee jiirka, oxycodone ayaa la barbar dhigay morphine oo muujiyay ka-hortagga ka-hortagga ka-hortagga dabada iyo saxanka kulul ka dib tabar-daran iyo ka-hortagnaan kooban.
Ka dib maamulka nidaamka (subcutaneous ama intraperitoneal), oxycodone ayaa lagu muujiyay in 2-4 jeer ka waxtar badan yahay morphine. Iibso Oxycodone Oxycontin 30mg online gudaha Australia
Natiijooyinkani waxay muujiyeen in dheef-shiid kiimikaadka firfircoon ee oxycodone (tusaale, oxymorphone) ay muhiim u noqon karaan xanuunka xanuunka dhexdhexaadka ah ee oxycodone. Daraasado la adeegsanayo jiirka Aguti mugdiga ah ee ku yar enzyme CYP2D1, kaas oo looga baahan yahay O-demethylate oxycodone ee jiirka, iyo antagonists kala duwan oo opioid ah ayaa soo jeediyay in antinociceptive Saamaynta oxycodone waxay noqon kartaa κ-opioid reseptor-dhexdhexaadin.
Faallooyin
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