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Oxycodone yanga iri mukushandiswa kwekiriniki kubvira 1917. Tenga Oxycodone Oxycontin 30mg online muAustralia.
Yakapihwa kuvanhu netsinga (iv),
intramuscularly (im),
intranasally (mu),
subcutaneously (sc),
chokwadi,
epidurally,
uye nemuromo uchishandisa zvigadziriso zvinokurumidza kuburitswa, uye mahwendefa ekukurumidza uye anodzorwa. Tenga Oxycodone Oxycontin 30mg online muAustralia
Iyo transdermal nzira yekutonga yakaedzwa zvakare mumhuka.
Nhoroondo | Oxycontin yePain Management | Mushroomifi.
Yakashandiswa kuchamhembe kweEurope kunyanya kurwadziwa kwakanyanya. MuCanada, Australia, uye United States, yainyanya kushandiswa semusanganiswa wemishonga ine acetaminophen, phenacetin, uye caffeine pakurwadziwa kuri pakati nepakati. MuFinland, oxycodone yakashandiswa seyakanyanya parenteral opioid yekurwadziwa kwakanyanya kubva kuma1960s. Tenga Oxycodone Oxycontin 30mg online muAustralia.
Chemistry uye Basic Pharmacology | OxyContin 30 mg mapiritsi ekuburitsa kwenguva refu | Mushroomifi.
-opioid receptor. Tenga Oxycodone Oxycontin 30mg online muAustralia
Iyo μ-opioid receptor inosunga hukama hweoxycodone, zvisinei, ishoma pane iyo yemorphine kana methadone.
Oxymorphone, iyo inoshanda metabolite yeoxycodone, ine yakanyanya kukwirira μ-opioid receptor inosunga hukama.
Intramuscular oxymorphone uye morphine yakaenzaniswa nevarwere vane kurwadziwa kusingaperi nekuda kwekenza. Intramuscular oxymorphone yakaratidza kuva 8.7 nguva dzine simba se morphine maererano nehuwandu hweanalgesic effect uye 13 nguva seine simba maererano nepamusoro pekuita.
Muzvidzidzo zvekuzvibata mumakonzo, oxycodone yakafananidzwa na Morphine uye yakaratidza zvakanyanya kusimba uye kupfupisa antinociception mumuswe flick uye inopisa ndiro bvunzo mushure me intrathecal (iyo) uye intracerebroventricular (icv) kutonga.
Mushure mekuita systemic administration (subcutaneous kana intraperitoneal), oxycodone yakaratidzwa kuva 2-4 nguva yakawanda kupfuura morphine. Tenga Oxycodone Oxycontin 30mg online muAustralia
Mhedzisiro iyi yakaratidza kuti iyo inoshanda metabolites yeoxycodone (semuenzaniso, oxymorphone) inogona kuve yakakosha mune oxycodone-mediated analgesia. Zvidzidzo zvinoshandisa Rima Aguti makonzo ayo asina kukwana mu enzyme CYP2D1, inodiwa kuO-demethylate oxycodone mugonzo, uye akasiyana maopioid receptor anopikisa akataura kuti antinociceptive Migumisiro ye oxycodone inogona kuva κ-opioid receptor-mediated.
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