SIYAN OXYCODONE 30MG X 100 KWALALA ONLINE | MUSHROOMIFI
Oxycodone yana cikin amfani na asibiti tun 1917. Sayi Oxycodone Oxycontin 30mg akan layi a Ostiraliya
An ba da shi ga ɗan adam ta hanyar jijiya (iv),
intramuscularly (im),
intrasally (cikin ciki),
subcutaneously (sc),
kai tsaye,
epiduraly,
da baki ta hanyar amfani da mafita-sakin-nan da nan, da allunan-saki-nan da nan da sarrafawa. Sayi Oxycodone Oxycontin 30mg akan layi a Ostiraliya
Hakanan an gwada hanyar da za a bi ta hanyar gudanarwa a cikin dabbobi.
Tarihi | Oxycontin don Gudanar da Raɗaɗi | Naman kaza.
An yi amfani da shi a arewacin Turai musamman don ciwo mai tsanani. A cikin Kanada, Ostiraliya, da Amurka, an yi amfani da shi musamman azaman maganin haɗin gwiwa tare da acetaminophen, phenacetin, da maganin kafeyin don matsakaicin zafi. A Finland, an yi amfani da oxycodone a matsayin babban opioid parenteral don ciwo mai tsanani tun daga 1960s. Sayi Oxycodone Oxycontin 30mg akan layi a Ostiraliya.
Chemistry da Basic Pharmacology | OxyContin 30 MG Allunan saki na tsawon lokaci | Naman kaza.
- mai karɓa na opioid. Sayi Oxycodone Oxycontin 30mg akan layi a Ostiraliya
Dangantakar mai karɓar μ-opioid na oxycodone shine, duk da haka, ƙasa da na morphine ko methadone.
Oxymorphone, metabolite mai aiki na oxycodone, yana da kusancin mai karɓa na μ-opioid mafi girma.
Intramuscular oxymorphone da morphine an kwatanta su a cikin marasa lafiya da ciwo mai tsanani saboda ciwon daji. Oxymorphone intramuscular ya tabbatar da cewa yana da ƙarfi sau 8.7 kamar morphine dangane da jimlar tasirin analgesic da sau 13 a matsayin mai ƙarfi dangane da tasirin kololuwa.
A cikin nazarin halaye a cikin berayen, Kwayoyin oxygen an kwatanta da morphine kuma ya nuna rashin ƙarfi da taƙaitaccen antinociception a cikin wutsiya flick da gwajin farantin zafi bayan intrathecal (shi) da intracerebroventricular (icv).
Bayan tsarin tsarin (subcutaneous ko intraperitoneal), an nuna oxycodone ya zama sau 2-4 mafi tasiri fiye da morphine. Sayi Oxycodone Oxycontin 30mg akan layi a Ostiraliya
Waɗannan sakamakon sun nuna cewa ƙwayoyin metabolites masu aiki na oxycodone (misali, oxymorphone) na iya zama mahimmanci a cikin analgesia mai tsaka-tsakin oxycodone. Nazarin da aka yi amfani da berayen Dark Aguti waɗanda ke da kasawa a cikin enzyme CYP2D1, wanda ake buƙata don O-demethylate oxycodone a cikin bera, da antagonists masu karɓar karɓar opioid daban-daban sun ba da shawarar cewa antinociceptive Tasirin oxycodone na iya zama κ-opioid mai karɓa-mai shiga tsakani.
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